Arimidex Anastrozole raw powder

Mifepristone Anti Estrogen Steroids Anastrozole / Arimidex Powder CAS 120511-73-1

Arimidex is a drug used to treat breast cancer in post-menopausal women (women who have gone through the menopause/ change of life).

It is a type of hormone treatment known as an aromatase inhibitor. The female hormone oestrogen stimulates some breast cancers to grow. These are described as hormone sensitive or receptor positive tumours.

Arimidex Usage: in Building Muscle, Burning Fat and Gaining Streng

Items Standard Results
Description White crystalline powder Complies
Identification IR
HPLC
Reactive
Conform with standard IR
Conform with standard HPLC
Conform
Solubility Freely soluble in methanol,acetone,
ethanol and tetrahydrofuran.
And very soluble in acetonitrile
Complies
Total Impurity max.0.5% 0.18%
Total Unspecified Impurity max. 0.2% 0.08%
Individual unspecified impurlty max. 0.1% 0.05%
Related compound B max. 0.2% 0.07%
Related compound C max. 0.2% 0.04%
Related compound D max. 0.1% 0.05%
Related compound E max. 0.1% 0.06%
Limit of cyclohexane max. 0.08% ND
Limit of ethylacetate max. 0.1% 0.07%
Melting point 81.0~84.0潞C 82.5~83.2潞C
Water max. 0.3% 0.21%
Residue on ignition max. 0.1% 0.07%
Heavy Metals max.0.001% Complies
Assay(HPLC) 98.0%~102.0% 99.8%
Storage Cool and dry
Conclusion It complies to USP32 .

Post-menopausal women do continue to produce oestrogen.This is mostly produced when other hormones are converted into oestrogen by an enzyme known as aromatase, which is found in the liver and the fatty tissues of the body.

Arimidex works by stopping this conversion from taking place so that the amount of oestrogen circulating in the body is reduced.

Anastrozole has been tested for reducing estrogens, including estradiol, in men.Excess estradiol in men can cause benign prostatic hyperplasia, gynecomastia, and symptoms of hypogonadism.

It can also contribute to increased risk of stroke, heart attack, chronic inflammation, prostate enlargement and prostate cancer.

Some athletes and body builders use anastrozole as part of their steroid cycle to reduce and prevent symptoms of excess estrogen-gynecomastia, emotional lability and water retention.

Arimidex Dosage:

This is a very potent drug that prevents the body from converting testosterone into estrogen. The drawback is that is very expensive. The minimum effective dosage is around between a quarter and a half of a milligram/day.

This drug does not need to be combined with any other during the cycle; however I recommend you begin using arimidex two weeks prior to commencing your cycle so that the drug can effectively eliminate the enzyme that permits conversion of testosterone to estrogen.

Arimidex Liquid Recipe:

Nolvadex:

Highest concentration made – 20mg/ml

Per 1 gram of Tamoxifen Citrate you will need:

9.8 ml’s of PEG 600

39.2 ml’s of 190 Proof Grain Alcohol

Armidex:

Highest concentration made – 5mg/ml

19.9 ml’s PEG 300

179.1 ml’s of 190 Proof Grain Alcohol

Clomid:

Highest concentration made – 50mg/ml

Per 1 gram of Clomiphene Citrate you will need:

8.4 ml’s of PEG 600

10.5 ml’s 190 Proof Grain Alcohol

Femara:

Highest concentration made – 5mg/ml

19.9 ml’s PEG 300

179.1 ml’s of 190 Proof Grain Alcohol

Product Name Arimidex
CAS 120511-73-4
Molecular Formula C17H19N5
Molecular Weight 293.37
Melting Point 81.0~84.0ºC
Assay 99.5%
Appearance White powder

How Arimidex Works:

Hormones are chemical substances that are produced by glands in the body, which enter the bloodstream and cause effects in other tissues.

For example, the hormone testosterone made in the testicles and is responsible for male characteristics such as deepening voice and increased body hair.

The use of hormone therapy to treat cancer is based on the observation that receptors for specific hormones that are needed for cell growth are on the surface of some tumor cells.

Hormone therapies work by stopping the production of a certain hormone, blocking hormone receptors, or substituting chemically similar agents for the active hormone, which cannot be used by the tumor cell.

The different types of hormone therapies are categorized by their function and/or the type of hormone that is effected.

Arimidex is an aromatase inhibitor. This means it blocks the enzyme aromatase (found in the body’s muscle, skin, breast and fat),

which is used to convert androgens (hormones produced by the adrenal glands) into estrogen. In the absence of estrogen, tumors dependent on this hormone for growth will shrink.  

Arimidex (Anastrozole) is the Aromatase inhibitor of choice. Arimidex’s mechanism of action – blocking conversion of Aromatizable steroids to estrogen – is in contrast to the mechanism of action of anti-estrogens,

such as Clomiphene (Clomid) or Tamoxifen (Nolvadex), which block estrogen receptors in some tissues, and activate estrogen receptors in others.

The drug is appropriately used when using substantial amounts of aromatizing steroids, or when one is prone to Gynecomastia and using moderate amounts of such steroids.

Arimidex does not have the side effects of Aminoglutethimide (Cytadren) and can achieve a high degree of estrogen blockade, much more than Cytadren.

It is possible to reduce estrogen too much with Arimidex, and for this reason, blood tests, or less preferably salivary tests, should be taken after the first week of use to determine if the dosage is correct.

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